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Natural product inspired optimization of a selective TRPV6 calcium channel inhibitor

Transient receptor potential vanilloid 6 (TRPV6) is a calcium channel implicated in multifactorial diseases and overexpressed in numerous cancers. We recently reported the phenyl-cyclohexyl-piperazine cis-22a as the first submicromolar TRPV6 inhibitor. This inhibitor showed a seven-fold selectivity...

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Detalhes bibliográficos
Publicado no:RSC Med Chem
Main Authors: Cunha, Micael Rodrigues, Bhardwaj, Rajesh, Carrel, Aline Lucie, Lindinger, Sonja, Romanin, Christoph, Parise-Filho, Roberto, Hediger, Matthias A., Reymond, Jean-Louis
Formato: Artigo
Idioma:Inglês
Publicado em: Royal Society of Chemistry 2020
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7513592/
https://ncbi.nlm.nih.gov/pubmed/33479695
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/d0md00145g
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