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Improved scale-up synthesis and purification of clinical asthma candidate MIDD0301

We report an improved and scalable synthesis of MIDD0301, a positive GABA(A) receptor modulator that is under development as oral and inhaled treatments for asthma. In contrast to other benzodiazepines in clinical use, MIDD0301 is a chiral compound that has limited brain absorption. The starting mat...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Org Process Res Dev
Hauptverfasser: Knutson, Daniel E., Roni, Rashid, Mian, Yeunus, Cook, James M., Stafford, Douglas C., Arnold, Leggy A.
Format: Artigo
Sprache:Inglês
Veröffentlicht: 2020
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC7497793/
https://ncbi.nlm.nih.gov/pubmed/32952391
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.oprd.0c00200
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