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Identification of a New Allosteric Binding Site for Cocaine in Dopamine Transporter

Dopamine (DA) transporter (DAT) is a major target for psychostimulant drugs of abuse such as cocaine that competitively binds to DAT, inhibits DA reuptake, and consequently increases synaptic DA levels. In addition to the central binding site inside DAT, the available experimental evidence suggests...

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Publicat a:J Chem Inf Model
Autors principals: Xu, Liang, Chen, Liao Y.
Format: Artigo
Idioma:Inglês
Publicat: 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7484383/
https://ncbi.nlm.nih.gov/pubmed/32649824
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.0c00346
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