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The Necessity of Using Changes in Absorption Time to Implicate Intestinal Transporter Involvement in Oral Drug-Drug Interactions

INTRODUCTION: In drug discovery and development, it is of high interest to characterize the potential for intestinal drug-drug interactions to alter bioavailability of a victim drug. For drugs that are substrates of both intestinal transporters and enzymes, estimating the relative contribution of ea...

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Dettagli Bibliografici
Pubblicato in:AAPS J
Autori principali: Sodhi, Jasleen K., Benet, Leslie Z.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7478332/
https://ncbi.nlm.nih.gov/pubmed/32808084
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1208/s12248-020-00469-6
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