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Simple binding of protein kinase A prior to phosphorylation allows CFTR anion channels to be opened by nucleotides

The Cystic Fibrosis Transmembrane Conductance Regulator (CFTR) anion channel is essential for epithelial salt–water balance. CFTR mutations cause cystic fibrosis, a lethal incurable disease. In cells CFTR is activated through the cAMP signaling pathway, overstimulation of which during cholera leads...

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Publicado en:Proc Natl Acad Sci U S A
Autores principales: Mihályi, Csaba, Iordanov, Iordan, Töröcsik, Beáta, Csanády, László
Formato: Artigo
Lenguaje:Inglês
Publicado: National Academy of Sciences 2020
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7474675/
https://ncbi.nlm.nih.gov/pubmed/32817533
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.2007910117
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