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Thrombospondin-1 counteracts the p97 inhibitor CB-5083 in colon carcinoma cells

p97 has recently emerged as a therapeutic target for cancer due to its essential functions in protein homeostasis. CB-5083 is a first-in-class, potent and selective ATP-competitive p97 inhibitor that induces proteotoxic stress in cancer cells. Potential mechanisms regulating the sensitivity of cells...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Cell Cycle
Egile Nagusiak: Her, Nam-Gu, Kesari, Santosh, Nurmemmedov, Elmar
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: Taylor & Francis 2020
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC7469669/
https://ncbi.nlm.nih.gov/pubmed/32423265
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/15384101.2020.1754584
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