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Structural Basis of p97 Inhibition by the Site-Selective Anticancer Compound CB-5083

Inhibition of p97, a key player in the ubiquitin-proteasome degradation pathway, has been proposed as a treatment of cancer. This concept was nearly realized recently when a potent p97 inhibitor, 1-[4-(benzylamino)-5H,7H,8H-pyrano[4,3-d]pyrimidin-2-yl]-2-methyl-1H-indole-4-carboxamide (CB-5083), was...

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Detalhes bibliográficos
Publicado no:Mol Pharmacol
Main Authors: Tang, Wai Kwan, Odzorig, Taivan, Jin, Whitney, Xia, Di
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6355941/
https://ncbi.nlm.nih.gov/pubmed/30591537
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.118.114256
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