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Structure-based evolution of a promiscuous inhibitor to a selective stabilizer of protein–protein interactions

The systematic stabilization of protein–protein interactions (PPI) has great potential as innovative drug discovery strategy to target novel and hard-to-drug protein classes. The current lack of chemical starting points and focused screening opportunities limits the identification of small molecule...

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Vydáno v:Nat Commun
Hlavní autoři: Sijbesma, Eline, Visser, Emira, Plitzko, Kathrin, Thiel, Philipp, Milroy, Lech-Gustav, Kaiser, Markus, Brunsveld, Luc, Ottmann, Christian
Médium: Artigo
Jazyk:Inglês
Vydáno: Nature Publishing Group UK 2020
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7414219/
https://ncbi.nlm.nih.gov/pubmed/32770072
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41467-020-17741-0
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