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Putative mGluR4 Positive Allosteric Modulators Activate G(i)-Independent Anti-Inflammatory Mechanisms in Microglia

Chronic dysregulated microglial activation may lead to persistent inflammation and progressive neurodegeneration. A previous study reported that ADX88178, a putative metabotropic glutamate receptor 4 (mGluR4) positive allosteric modulator (PAM), exerts anti-inflammatory effects in microglia by activ...

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Detalles Bibliográficos
Publicado en:Neurochem Int
Autores principales: Abulwerdi, Gelareh, Stoica, Bogdan A., Loane, David J., Faden, Alan I.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2020
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7392812/
https://ncbi.nlm.nih.gov/pubmed/32454165
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuint.2020.104770
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