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Blocking EGFR palmitoylation suppresses PI3K signaling and mutant KRAS lung tumorigenesis

Nonsmall cell lung cancer (NSCLC) is often characterized by mutually exclusive mutations in the epidermal growth factor receptor (EGFR) or the guanosine triphosphatase KRAS. We hypothesized that blocking EGFR palmitoylation, previously shown to inhibit EGFR activity, might alter downstream signaling...

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Pubblicato in:Sci Signal
Autori principali: Kharbanda, Akriti, Walter, David, Guidel, Andrea, Schek, Nancy, Feldser, David, Witze, Eric S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7310254/
https://ncbi.nlm.nih.gov/pubmed/32127496
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/scisignal.aax2364
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