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MARCH5 mediates NOXA-dependent MCL1 degradation driven by kinase inhibitors and integrated stress response activation

MCL1 has critical antiapoptotic functions and its levels are tightly regulated by ubiquitylation and degradation, but mechanisms that drive this degradation, particularly in solid tumors, remain to be established. We show here in prostate cancer cells that increased NOXA, mediated by kinase inhibito...

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Publicat a:eLife
Autors principals: Arai, Seiji, Varkaris, Andreas, Nouri, Mannan, Chen, Sen, Xie, Lisha, Balk, Steven P
Format: Artigo
Idioma:Inglês
Publicat: eLife Sciences Publications, Ltd 2020
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7297531/
https://ncbi.nlm.nih.gov/pubmed/32484436
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.7554/eLife.54954
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