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Small molecule H89 renders the phosphorylation of S6K1 and AKT resistant to mTOR inhibitors

The mammalian target of rapamycin (mTOR) is an evolutionarily conserved Ser/Thr kinase that comprises two complexes, termed mTOR complex 1 (mTORC1) and mTOR complex 2 (mTORC2). mTORC1 phosphorylates S6K1 at Thr 389, whereas mTORC2 phosphorylates AKT at Ser 473 to promote cell growth. As the mTOR nam...

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Bibliografske podrobnosti
izdano v:Biochem J
Main Authors: Melick, Chase H., Jewell, Jenna L.
Format: Artigo
Jezik:Inglês
Izdano: Portland Press Ltd. 2020
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC7261416/
https://ncbi.nlm.nih.gov/pubmed/32347294
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BCJ20190958
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