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IACS-010759, a potent inhibitor of glycolysis-deficient hypoxic tumor cells, inhibits mitochondrial respiratory complex I through a unique mechanism

The small molecule IACS-010759 has been reported to potently inhibit the proliferation of glycolysis-deficient hypoxic tumor cells by interfering with the functions of mitochondrial NADH-ubiquinone oxidoreductase (complex I) without exhibiting cytotoxicity at tolerated doses in normal cells. Conside...

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Dettagli Bibliografici
Pubblicato in:J Biol Chem
Autori principali: Tsuji, Atsuhito, Akao, Takumi, Masuya, Takahiro, Murai, Masatoshi, Miyoshi, Hideto
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Biochemistry and Molecular Biology 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7247293/
https://ncbi.nlm.nih.gov/pubmed/32295842
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA120.013366
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