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Discovery of Novel Pyrazolo-Pyridone DCN1 Inhibitors Controlling Cullin Neddylation

Chemical control of cullin neddylation is attracting increased attention based largely on the successes of the NEDD8-activating enzyme (E1) inhibitor Pevonedistat. Recently reported chemical probes enable selective and time-dependent inhibition of downstream members of the neddylation tri-enzymatic...

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Vydáno v:J Med Chem
Hlavní autoři: Kim, Ho Shin, Hammill, Jared T., Scott, Daniel C., Chen, Yizhe, Min, Jaeki, Rector, Jonah, Singh, Bhuvanesh, Schulman, Brenda A., Guy, R. Kiplin
Médium: Artigo
Jazyk:Inglês
Vydáno: 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7228038/
https://ncbi.nlm.nih.gov/pubmed/31465221
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.9b00410
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