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Computer-Driven Development of an in Silico Tool for Finding Selective Histone Deacetylase 1 Inhibitors
Histone deacetylases (HDACs) are a class of epigenetic modulators overexpressed in numerous types of cancers. Consequently, HDAC inhibitors (HDACIs) have emerged as promising antineoplastic agents. Unfortunately, the most developed HDACIs suffer from poor selectivity towards a specific isoform, limi...
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| Publicat a: | Molecules |
|---|---|
| Autors principals: | , , , , |
| Format: | Artigo |
| Idioma: | Inglês |
| Publicat: |
MDPI
2020
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| Matèries: | |
| Accés en línia: | https://ncbi.nlm.nih.gov/pmc/articles/PMC7221830/ https://ncbi.nlm.nih.gov/pubmed/32331470 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules25081952 |
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