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Semimechanistic Modeling to Guide Venetoclax Coadministration with Ritonavir and Digoxin

Venetoclax is a cytochrome P450, family 3, subfamily A (CYP3A) substrate and was shown to inhibit P‐gp efflux transporters in vitro. To quantify the impact of CYP3A inhibition by ritonavir on venetoclax disposition and P‐gp inhibition by venetoclax on digoxin pharmacokinetics, two semimechanistic dr...

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Detalhes bibliográficos
Publicado no:Clin Transl Sci
Main Authors: Alhadab, Ali A., Salem, Ahmed Hamed, Freise, Kevin J.
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2020
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7214649/
https://ncbi.nlm.nih.gov/pubmed/31961475
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/cts.12739
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