Učitavanje...

Thiol-Reactive PODS-Bearing Bifunctional Chelators for the Development of EGFR-Targeting [(18)F]AlF-Affibody Conjugates

Site-selective bioconjugation of cysteine-containing peptides and proteins is currently achieved via a maleimide–thiol reaction (Michael addition). When maleimide-functionalized chelators are used and the resulting bioconjugates are subsequently radiolabeled, instability has been observed both durin...

Cijeli opis

Spremljeno u:
Bibliografski detalji
Izdano u:Molecules
Glavni autori: Da Pieve, Chiara, Makarem, Ata, Turnock, Stephen, Maczynska, Justyna, Smith, Graham, Kramer-Marek, Gabriela
Format: Artigo
Jezik:Inglês
Izdano: MDPI 2020
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC7180749/
https://ncbi.nlm.nih.gov/pubmed/32235296
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules25071562
Oznake: Dodaj oznaku
Bez oznaka, Budi prvi tko označuje ovaj zapis!