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TBAJ-876, a 3,5-Dialkoxypyridine Analogue of Bedaquiline, Is Active against Mycobacterium abscessus

Lung disease caused by Mycobacterium abscessus is very difficult to cure, and treatment failure rates are high. The antituberculosis drug bedaquiline (BDQ) is used as salvage therapy against this dreadful disease. However, BDQ is highly lipophilic, displays a long terminal half-life, and presents a...

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Detalles Bibliográficos
Publicado en:Antimicrob Agents Chemother
Main Authors: Sarathy, Jickky Palmae, Ganapathy, Uday S., Zimmerman, Matthew D., Dartois, Véronique, Gengenbacher, Martin, Dick, Thomas
Formato: Artigo
Idioma:Inglês
Publicado: American Society for Microbiology 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7179298/
https://ncbi.nlm.nih.gov/pubmed/31964791
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.02404-19
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