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Strategies for developing pregnane X receptor antagonists: Implications from metabolism to cancer

Pregnane X receptor (PXR) is a ligand-activated nuclear receptor that was originally identified as a master regulator of xenobiotic detoxification. It regulates the expression of drug-metabolizing enzymes and transporters to control the degradation and excretion of endobiotics and xenobiotics, inclu...

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Dettagli Bibliografici
Pubblicato in:Med Res Rev
Autori principali: Chai, Sergio C., Wright, William C., Chen, Taosheng
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC7166136/
https://ncbi.nlm.nih.gov/pubmed/31782213
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/med.21648
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