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Allosteric GABA(A) Receptor Modulators—A Review on the Most Recent Heterocyclic Chemotypes and Their Synthetic Accessibility †

GABA(A) receptor modulators are structurally almost as diverse as their target protein. A plethora of heterocyclic scaffolds has been described as modulating this extremely important receptor family. Some made it into clinical trials and, even on the market, some were dismissed. This review focuses...

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Publicado en:Molecules
Main Authors: Vega Alanis, Blanca Angelica, Iorio, Maria Teresa, Silva, Luca L., Bampali, Konstantina, Ernst, Margot, Schnürch, Michael, Mihovilovic, Marko D.
Formato: Artigo
Idioma:Inglês
Publicado: MDPI 2020
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC7070463/
https://ncbi.nlm.nih.gov/pubmed/32102309
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules25040999
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