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Sequence and structural determinants of ligand-dependent alternating access of a MATE transporter

Multidrug and toxic compound extrusion (MATE) transporters are ubiquitous ion-coupled antiporters that extrude structurally and chemically dissimilar cytotoxic compounds and have been implicated in conferring multidrug resistance. Here, we integrate double electron–electron resonance (DEER) with fun...

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Detalles Bibliográficos
Publicado en:Proc Natl Acad Sci U S A
Autores principales: Jagessar, Kevin L., Claxton, Derek P., Stein, Richard A., Mchaourab, Hassane S.
Formato: Artigo
Lenguaje:Inglês
Publicado: National Academy of Sciences 2020
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC7060674/
https://ncbi.nlm.nih.gov/pubmed/32075917
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.1917139117
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