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Brain Distributional Kinetics of a Novel MDM2 Inhibitor SAR405838: Implications for Use in Brain Tumor Therapy

Achieving an effective drug concentration in the brain is as important as targeting the right pathway when developing targeted agents for brain tumors. SAR405838 is a novel molecularly targeted agent that is in clinical trials for various solid tumors. Its application for tumors in the brain has not...

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Detalhes bibliográficos
Publicado no:Drug Metab Dispos
Main Authors: Kim, Minjee, Laramy, Janice K., Gampa, Gautham, Parrish, Karen E., Brundage, Richard, Sarkaria, Jann N., Elmquist, William F.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2019
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC7042719/
https://ncbi.nlm.nih.gov/pubmed/31619389
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.119.088716
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