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Synthetic Approaches to Zetekitoxin AB, a Potent Voltage-Gated Sodium Channel Inhibitor

Voltage-gated sodium channels (Na(V)s) are membrane proteins that are involved in the generation and propagation of action potentials in neurons. Recently, the structure of a complex made of a tetrodotoxin-sensitive (TTX-s) Na(V) subtype with saxitoxin (STX), a shellfish toxin, was determined. STX p...

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Dades bibliogràfiques
Publicat a:Mar Drugs
Autors principals: Adachi, Kanna, Ishizuka, Hayate, Odagi, Minami, Nagasawa, Kazuo
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC7024329/
https://ncbi.nlm.nih.gov/pubmed/31888062
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md18010024
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