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GABA(A) Receptor Ligands Often Interact with Binding Sites in the Transmembrane Domain and in the Extracellular Domain—Can the Promiscuity Code Be Cracked?

Many allosteric binding sites that modulate gamma aminobutyric acid (GABA) effects have been described in heteropentameric GABA type A (GABA(A)) receptors, among them sites for benzodiazepines, pyrazoloquinolinones and etomidate. Diazepam not only binds at the high affinity extracellular “canonical”...

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Detaylı Bibliyografya
Yayımlandı:Int J Mol Sci
Asıl Yazarlar: Iorio, Maria Teresa, Vogel, Florian Daniel, Koniuszewski, Filip, Scholze, Petra, Rehman, Sabah, Simeone, Xenia, Schnürch, Michael, Mihovilovic, Marko D., Ernst, Margot
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: MDPI 2020
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6982053/
https://ncbi.nlm.nih.gov/pubmed/31947863
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms21010334
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