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Comparative pharmacokinetics and pharmacodynamics of the advanced Retinol-Binding Protein 4 antagonist in dog and cynomolgus monkey

Accumulation of lipofuscin bisretinoids in the retina contributes to pathogenesis of macular degeneration. Retinol-Binding Protein 4 (RBP4) antagonists reduce serum retinol concentrations thus partially reducing retinol delivery to the retina which decreases bisretinoid synthesis. BPN-14136 is a nov...

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Pubblicato in:PLoS One
Autori principali: Racz, Boglarka, Varadi, Andras, Pearson, Paul G., Petrukhin, Konstantin
Natura: Artigo
Lingua:Inglês
Pubblicazione: Public Library of Science 2020
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6980506/
https://ncbi.nlm.nih.gov/pubmed/31978148
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0228291
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