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Pharmacokinetics and Safety of Single-Dose Esaxerenone in Japanese Subjects with Mild to Moderate Hepatic Impairment

INTRODUCTION: The mineralocorticoid receptor (MR) blocker esaxerenone is a new treatment for hypertension in Japan and under development for treatment of diabetic nephropathy. Hepatic impairment is known to impact the pharmacokinetics (PKs) of other MR blocking drugs. The aim of the present study wa...

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Bibliografski detalji
Izdano u:Adv Ther
Glavni autori: Kurata, Akifumi, Yoshida, Takafumi, Inoue, Megumi, Ishizuka, Tomoko, Nakatsu, Takafumi, Shimizu, Takako, Kato, Manabu, Nishikawa, Yasuhiro, Ishizuka, Hitoshi
Format: Artigo
Jezik:Inglês
Izdano: Springer Healthcare 2019
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6979450/
https://ncbi.nlm.nih.gov/pubmed/31705436
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s12325-019-01121-2
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