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NanoBiT Complementation to Monitor Agonist-Induced Adenosine A(1) Receptor Internalization

Receptor internalization in response to prolonged agonist treatment is an important regulator of G protein–coupled receptor (GPCR) function. The adenosine A(1) receptor (A(1)AR) is one of the adenosine receptor family of GPCRs, and evidence for its agonist-induced internalization is equivocal. The r...

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Dades bibliogràfiques
Publicat a:SLAS Discov
Autors principals: Soave, Mark, Kellam, Barrie, Woolard, Jeanette, Briddon, Stephen J., Hill, Stephen J.
Format: Artigo
Idioma:Inglês
Publicat: SAGE Publications 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6974774/
https://ncbi.nlm.nih.gov/pubmed/31583945
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1177/2472555219880475
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