Carregant...

Engineering Chemoselectivity in Hemoprotein-Catalyzed Indole Amidation

Here we report a cytochrome P450 variant that catalyzes C(2)-amidation of 1-methylindoles with tosyl azide via nitrene transfer. Before evolutionary optimization the enzyme exhibited two undesired side reactivities resulting in reduction of the putative iron-nitrenoid intermediate or cycloaddition b...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:ACS Catal
Autors principals: Brandenberg, Oliver F., Miller, David C., Markel, Ulrich, Chaib, Anissa Ouald, Arnold, Frances H.
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6959474/
https://ncbi.nlm.nih.gov/pubmed/31938573
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acscatal.9b02508
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!