A carregar...

Imidazolidine-2,4,5- and pirimidine-2,4,6-triones – new primary pharmacophore for soluble epoxide hydrolase inhibitors with enhanced water solubility.

A series of inhibitors of the soluble epoxide hydrolase (sEH) containing imidazolidine-2,4,5-trione or pirimidine-2,4,6-trione has been synthesized. Inhibition potency of the described compounds ranges from 8.4 μM to 0.4 nM. The tested compounds possess higher water solubility than their preceding u...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Burmistrov, Vladimir, Morisseau, Christophe, D’yachenko, Vladimir, Karlov, Dmitry, Butov, Gennady M., Hammock, Bruce D.
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6957307/
https://ncbi.nlm.nih.gov/pubmed/31870649
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2019.126908
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!