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Identification of C-6 as a New Site for Linker Conjugation to the Taccalonolide Microtubule Stabilizers

The taccalonolides are a class of microtubule stabilizers that circumvent clinically relevant forms of drug resistance due to their unique mechanism of microtubule stabilization imparted by the covalent binding of the C-22−–-23 epoxide moiety to tubulin. A taccalonolide (8) with a fluorescein group...

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Bibliografske podrobnosti
izdano v:J Nat Prod
Main Authors: Du, Lin, Risinger, April L., Yee, Samantha S., Ola, Antonius R. B., Zammiello, Cynthia L, Cichewicz, Robert H., Mooberry, Susan L.
Format: Artigo
Jezik:Inglês
Izdano: 2019
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6952213/
https://ncbi.nlm.nih.gov/pubmed/30799622
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jnatprod.8b01036
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