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Surface plasmon resonance and cytotoxicity assays of drug efficacies predicted computationally to inhibit p53/MDM2 interaction

Docking on the p53-binding site of murine double minute 2 (MDM2) by small molecules restores p53’s tumor-suppressor function. We previously assessed 3244 FDA-approved drugs via “computational conformer selection” for inhibiting MDM2 and p53 interaction. Here, we developed a surface plasmon resonance...

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Vydáno v:Anal Biochem
Hlavní autoři: Wang, Xiaoying, Magdziarz, Patrycja, Enriquez, Ernest, Zhao, Wang, Quan, Chris, Darabedian, Narek, Momand, Jamil, Zhou, Feimeng
Médium: Artigo
Jazyk:Inglês
Vydáno: 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6942878/
https://ncbi.nlm.nih.gov/pubmed/30721669
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ab.2019.01.012
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