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Lercanidipine Synergistically Enhances Bortezomib Cytotoxicity in Cancer Cells via Enhanced Endoplasmic Reticulum Stress and Mitochondrial Ca(2+) Overload

The proteasome inhibitor (PI), bortezomib (Btz), is effective in treating multiple myeloma and mantle cell lymphoma, but not solid tumors. In this study, we show for the first time that lercanidipine (Ler), an antihypertensive drug, enhances the cytotoxicity of various PIs, including Btz, carfilzomi...

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Detalles Bibliográficos
Publicado en:Int J Mol Sci
Autores principales: Lee, A Reum, Seo, Min Ji, Kim, Jin, Lee, Dong Min, Kim, In Young, Yoon, Mi Jin, Hoon, Hur, Choi, Kyeong Sook
Formato: Artigo
Lenguaje:Inglês
Publicado: MDPI 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6941136/
https://ncbi.nlm.nih.gov/pubmed/31817163
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20246112
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