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Lercanidipine Synergistically Enhances Bortezomib Cytotoxicity in Cancer Cells via Enhanced Endoplasmic Reticulum Stress and Mitochondrial Ca(2+) Overload

The proteasome inhibitor (PI), bortezomib (Btz), is effective in treating multiple myeloma and mantle cell lymphoma, but not solid tumors. In this study, we show for the first time that lercanidipine (Ler), an antihypertensive drug, enhances the cytotoxicity of various PIs, including Btz, carfilzomi...

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Dettagli Bibliografici
Pubblicato in:Int J Mol Sci
Autori principali: Lee, A Reum, Seo, Min Ji, Kim, Jin, Lee, Dong Min, Kim, In Young, Yoon, Mi Jin, Hoon, Hur, Choi, Kyeong Sook
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6941136/
https://ncbi.nlm.nih.gov/pubmed/31817163
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20246112
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