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Nutlin-3 enhances the bortezomib sensitivity of p53-defective cancer cells by inducing paraptosis

The proteasome inhibitor, bortezomib, is ineffective against many solid tumors. Nutlin-3 is a potent antagonist of human homolog of murine double minute 2/p53 interaction exhibiting promising therapeutic anti-cancer activity. In this study, we show that treatment of various p53-defective bortezomib-...

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Pubblicato in:Exp Mol Med
Autori principali: Lee, Dong Min, Kim, In Young, Seo, Min Ji, Kwon, Mi Ri, Choi, Kyeong Sook
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5579507/
https://ncbi.nlm.nih.gov/pubmed/28798402
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/emm.2017.112
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