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Trimerization of dopamine transporter triggered by AIM-100 binding: Molecular mechanism and effect of mutations

Recent work demonstrated the propensity of dopamine transporters (DATs) to form trimers or higher oligomers, enhanced upon binding a furopyrimidine, AIM-100. AIM-100 binding promotes DAT endocytosis and thereby moderates dopaminergic transmission. Despite the neurobiological significance of these ev...

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Pubblicato in:Neuropharmacology
Autori principali: Cheng, Mary Hongying, Ponzoni, Luca, Sorkina, Tatiana, Lee, Ji Young, Zhang, She, Sorkin, Alexander, Bahar, Ivet
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6917874/
https://ncbi.nlm.nih.gov/pubmed/31228486
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuropharm.2019.107676
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