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Targeted Protein Degradation by Chimeric Small Molecules, PROTACs and SNIPERs

Technologies that induce targeted protein degradation by small molecules have been developed recently. Chimeric small molecules such as Proteolysis Targeting Chimeras (PROTACs) and Specific and Non-genetic IAP-dependent Protein Erasers (SNIPERs), and E3 modulators such as thalidomides, hijack the ce...

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Detalles Bibliográficos
Publicado en:Front Chem
Main Authors: Naito, Mikihiko, Ohoka, Nobumichi, Shibata, Norihito, Tsukumo, Yoshinori
Formato: Artigo
Idioma:Inglês
Publicado: Frontiers Media S.A. 2019
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6914816/
https://ncbi.nlm.nih.gov/pubmed/31921772
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fchem.2019.00849
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