Wordt geladen...

Novel Lysine-Based Thioureas as Mechanism-Based Inhibitors of Sirtuin 2 (SIRT2) with Anticancer Activity in a Colorectal Cancer Murine Model

Sirtuin 2 (SIRT2) is a protein lysine deacylase that has been indicated as a therapeutic target for cancer. To further establish the role of SIRT2 in cancers, it is necessary to develop selective and potent inhibitors. Here, we report the facile synthesis of novel lysine derived thioureas as mechani...

Volledige beschrijving

Bewaard in:
Bibliografische gegevens
Gepubliceerd in:J Med Chem
Hoofdauteurs: Farooqi, Ali Sohail, Hong, Jun Young, Cao, Ji, Lu, Xuan, Price, Ian Robert, Zhao, Qingjie, Kosciuk, Tatsiana, Yang, Min, Bai, Jessica Jingyi, Lin, Hening
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2019
Onderwerpen:
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6901289/
https://ncbi.nlm.nih.gov/pubmed/30986062
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.9b00191
Tags: Voeg label toe
Geen labels, Wees de eerste die dit record labelt!