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Novel Lysine-Based Thioureas as Mechanism-Based Inhibitors of Sirtuin 2 (SIRT2) with Anticancer Activity in a Colorectal Cancer Murine Model

Sirtuin 2 (SIRT2) is a protein lysine deacylase that has been indicated as a therapeutic target for cancer. To further establish the role of SIRT2 in cancers, it is necessary to develop selective and potent inhibitors. Here, we report the facile synthesis of novel lysine derived thioureas as mechani...

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Vydáno v:J Med Chem
Hlavní autoři: Farooqi, Ali Sohail, Hong, Jun Young, Cao, Ji, Lu, Xuan, Price, Ian Robert, Zhao, Qingjie, Kosciuk, Tatsiana, Yang, Min, Bai, Jessica Jingyi, Lin, Hening
Médium: Artigo
Jazyk:Inglês
Vydáno: 2019
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On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6901289/
https://ncbi.nlm.nih.gov/pubmed/30986062
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.9b00191
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