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Recent Advances in Selective and Irreversible Covalent Ligand Development and Validation

Some of the most widely used drugs, like aspirin and penicillin, are covalent drugs. Covalent binding can improve potency, selectivity and duration of the effects, but the intrinsic reactivity represents a potential liability and may result in idiosyncratic toxicity. For decades, the cons were belie...

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Podrobná bibliografie
Vydáno v:Cell Chem Biol
Hlavní autoři: Zhang, Tinghu, Hatcher, John M., Teng, Mingxing, Gray, Nathanael S., Kostic, Milka
Médium: Artigo
Jazyk:Inglês
Vydáno: 2019
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6886688/
https://ncbi.nlm.nih.gov/pubmed/31631011
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.chembiol.2019.09.012
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