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Pharmacological and Molecular Mechanisms Behind the Sterilizing Activity of Pyrazinamide

Inclusion of pyrazinamide in the tuberculosis drug regimen in the 1970s allowed reduction of treatment duration from 12 to 6 months. Pyrazinamide has this remarkable effect in patients despite displaying poor potency against Mycobacterium tuberculosis in vitro. The pharmacological basis for the drug...

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Publicat a:Trends Pharmacol Sci
Autors principals: Gopal, Pooja, Grüber, Gerhard, Dartois, Véronique, Dick, Thomas
Format: Artigo
Idioma:Inglês
Publicat: 2019
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6884696/
https://ncbi.nlm.nih.gov/pubmed/31704175
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.tips.2019.10.005
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