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Identification of Candidate Risk Factor Genes for Human Idelalisib Toxicity Using a Collaborative Cross Approach

Idelalisib is a phosphatidylinositol 3-kinase inhibitor highly selective for the delta isoform that has shown good efficacy in treating chronic lymphocytic leukemia and follicular lymphoma. In clinical trials, however, idelalisib was associated with rare, but potentially serious liver and lung toxic...

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Dettagli Bibliografici
Pubblicato in:Toxicol Sci
Autori principali: Mosedale, Merrie, Cai, Yanwei, Eaddy, John Scott, Corty, Robert W, Nautiyal, Manisha, Watkins, Paul B, Valdar, William
Natura: Artigo
Lingua:Inglês
Pubblicazione: Oxford University Press 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6876541/
https://ncbi.nlm.nih.gov/pubmed/31501888
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/toxsci/kfz199
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