Cargando...
Prediction of Tissue-Plasma Partition Coefficients Using Microsomal Partitioning: Incorporation into Physiologically based Pharmacokinetic Models and Steady-State Volume of Distribution Predictions
Drug distribution is a necessary component of models to predict human pharmacokinetics. A new membrane-based tissue-plasma partition coefficient (K(p)) method (K(p,mem)) to predict unbound tissue to plasma partition coefficients (K(pu)) was developed using in vitro membrane partitioning [fraction un...
Guardado en:
| Publicado en: | Drug Metab Dispos |
|---|---|
| Autores principales: | , , , |
| Formato: | Artigo |
| Lenguaje: | Inglês |
| Publicado: |
The American Society for Pharmacology and Experimental Therapeutics
2019
|
| Materias: | |
| Acceso en línea: | https://ncbi.nlm.nih.gov/pmc/articles/PMC6750188/ https://ncbi.nlm.nih.gov/pubmed/31324699 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.119.087973 |
| Etiquetas: |
Agregar Etiqueta
Sin Etiquetas, Sea el primero en etiquetar este registro!
|