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Drug Distribution. Part 1. Models to Predict Membrane Partitioning

PURPOSE: Tissue partitioning is an important component of drug distribution and half-life. Protein binding and lipid partitioning together determine drug distribution. METHODS: Two structure-based models to predict partitioning into microsomal membranes are presented. An orientation-based model was...

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Publicado en:Pharm Res
Main Authors: Nagar, Swati, Korzekwa, Ken
Formato: Artigo
Idioma:Inglês
Publicado: 2016
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5588161/
https://ncbi.nlm.nih.gov/pubmed/27981450
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11095-016-2085-z
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