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One-step Heck Reaction Generates Nonimmunosuppressive FK506 Analogs for Pharmacological BMP Activation

[Image: see text] FKBP12 ligands such as FK506 have been shown to activate the BMP signaling pathway and facilitate tissue regeneration. However, the immunosuppressive activity of FK506 limits its clinical application. Using Heck reaction, we generated nonimmunosuppressive analogs of FK506 by fusing...

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Detalhes bibliográficos
Publicado no:ACS Med Chem Lett
Main Authors: Wang, Yuefan, Peiffer, Brandon J., Su, Qi, Liu, Jun O.
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2019
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6746090/
https://ncbi.nlm.nih.gov/pubmed/31531197
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.9b00144
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