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Biotransformation of the Mycotoxin Enniatin B1 by CYP P450 3A4 and Potential for Drug-Drug Interactions

Enniatins (ENNs) are fungal secondary metabolites that frequently occur in grain in temperate climates. Their toxic potency is connected to their ionophoric character and lipophilicity. The biotransformation of ENNs predominantly takes place via cytochrome P450 3A (CYP 3A)-dependent oxidation reacti...

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Detalhes bibliográficos
Publicado no:Metabolites
Main Authors: Ivanova, Lada, Denisov, Ilia G., Grinkova, Yelena V., Sligar, Stephen G., Fæste, Christiane K.
Formato: Artigo
Idioma:Inglês
Publicado em: MDPI 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6724072/
https://ncbi.nlm.nih.gov/pubmed/31357617
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/metabo9080158
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