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Ligand Binding Dynamics for Pre-dimerised G Protein-Coupled Receptor Homodimers: Linear Models and Analytical Solutions

Evidence suggests that many G protein-coupled receptors (GPCRs) are bound together forming dimers. The implications of dimerisation for cellular signalling outcomes, and ultimately drug discovery and therapeutics, remain unclear. Consideration of ligand binding and signalling via receptor dimers is...

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Publicat a:Bull Math Biol
Autors principals: White, Carla, Bridge, Lloyd J.
Format: Artigo
Idioma:Inglês
Publicat: Springer US 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6722261/
https://ncbi.nlm.nih.gov/pubmed/29349610
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11538-017-0387-x
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