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Ligand Binding Dynamics for Pre-dimerised G Protein-Coupled Receptor Homodimers: Linear Models and Analytical Solutions

Evidence suggests that many G protein-coupled receptors (GPCRs) are bound together forming dimers. The implications of dimerisation for cellular signalling outcomes, and ultimately drug discovery and therapeutics, remain unclear. Consideration of ligand binding and signalling via receptor dimers is...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:Bull Math Biol
Päätekijät: White, Carla, Bridge, Lloyd J.
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: Springer US 2018
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6722261/
https://ncbi.nlm.nih.gov/pubmed/29349610
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1007/s11538-017-0387-x
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