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Antinociceptive Activity of Thiazole-containing Cyclized DAMGO and Leu-(Met) Enkephalin Analogs

Numerous studies demonstrate the promise of opioid peptides as analgesics, but poor oral bioavailability has limited their therapeutic development. This study sought to increase the oral bioavailability of opioid peptides by cyclization, using Hantzsch-based macrocyclization strategies to produce tw...

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Detalhes bibliográficos
Publicado no:Org Biomol Chem
Main Authors: Harris, Hannah M., Eans, Shainnel O., Ganno, Michelle L., Davis, Jennifer C., Dooley, Colette T., McLaughlin, Jay P., Nefzi, Adel
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6637423/
https://ncbi.nlm.nih.gov/pubmed/31094391
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c9ob00882a
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