Cargando...

Productive reorientation of a bound oxime reactivator revealed in room temperature X-ray structures of native and VX-inhibited human acetylcholinesterase

Exposure to organophosphorus compounds (OPs) may be fatal if untreated, and a clear and present danger posed by nerve agent OPs has become palpable in recent years. OPs inactivate acetylcholinesterase (AChE) by covalently modifying its catalytic serine. Inhibited AChE cannot hydrolyze the neurotrans...

Descrición completa

Gardado en:
Detalles Bibliográficos
Publicado en:J Biol Chem
Main Authors: Gerlits, Oksana, Kong, Xiaotian, Cheng, Xiaolin, Wymore, Troy, Blumenthal, Donald K., Taylor, Palmer, Radić, Zoran, Kovalevsky, Andrey
Formato: Artigo
Idioma:Inglês
Publicado: American Society for Biochemistry and Molecular Biology 2019
Assuntos:
Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6615692/
https://ncbi.nlm.nih.gov/pubmed/31138650
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA119.008725
Tags: Engadir etiqueta
Sen Etiquetas, Sexa o primeiro en etiquetar este rexistro!