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Productive reorientation of a bound oxime reactivator revealed in room temperature X-ray structures of native and VX-inhibited human acetylcholinesterase

Exposure to organophosphorus compounds (OPs) may be fatal if untreated, and a clear and present danger posed by nerve agent OPs has become palpable in recent years. OPs inactivate acetylcholinesterase (AChE) by covalently modifying its catalytic serine. Inhibited AChE cannot hydrolyze the neurotrans...

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Библиографические подробности
Опубликовано в: :J Biol Chem
Главные авторы: Gerlits, Oksana, Kong, Xiaotian, Cheng, Xiaolin, Wymore, Troy, Blumenthal, Donald K., Taylor, Palmer, Radić, Zoran, Kovalevsky, Andrey
Формат: Artigo
Язык:Inglês
Опубликовано: American Society for Biochemistry and Molecular Biology 2019
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6615692/
https://ncbi.nlm.nih.gov/pubmed/31138650
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1074/jbc.RA119.008725
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