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Discovery of a Potent, Long‐Acting, and CNS‐Active Inhibitor (BIA 10‐2474) of Fatty Acid Amide Hydrolase

Fatty acid amide hydrolase (FAAH) can be targeted for the treatment of pain associated with various medical conditions. Herein we report the design and synthesis of a novel series of heterocyclic‐N‐carboxamide FAAH inhibitors that have a good alignment of potency, metabolic stability and selectivity...

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Shranjeno v:
Bibliografske podrobnosti
izdano v:ChemMedChem
Main Authors: Kiss, László E., Beliaev, Alexandre, Ferreira, Humberto S., Rosa, Carla P., Bonifácio, Maria João, Loureiro, Ana I., Pires, Nuno M., Palma, P. Nuno, Soares‐da‐Silva, Patrício
Format: Artigo
Jezik:Inglês
Izdano: John Wiley and Sons Inc. 2018
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6582431/
https://ncbi.nlm.nih.gov/pubmed/30113139
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cmdc.201800393
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